{"id":3602,"date":"2021-09-28T15:41:15","date_gmt":"2021-09-28T14:41:15","guid":{"rendered":"https:\/\/health-online-hero.com\/?p=3602"},"modified":"2024-03-01T18:43:30","modified_gmt":"2024-03-01T17:43:30","slug":"pfizer-unveils-oral-inhibitorpf-07321332-of-sars-cov-2-main-protease","status":"publish","type":"post","link":"https:\/\/health-online-hero.com\/en\/protection\/pfizer-unveils-oral-inhibitorpf-07321332-of-sars-cov-2-main-protease\/","title":{"rendered":"Pfizer unveils oral inhibitorPF-07321332 of SARS-CoV-2 main protease"},"content":{"rendered":"<p>[et_pb_section fb_built=&#8221;1&#8243; custom_padding_last_edited=&#8221;on|phone&#8221; admin_label=&#8221;Header&#8221; _builder_version=&#8221;4.8.1&#8243; use_background_color_gradient=&#8221;on&#8221; background_color_gradient_start=&#8221;rgba(255,255,255,0)&#8221; background_color_gradient_end=&#8221;#00a07a&#8221; background_color_gradient_overlays_image=&#8221;on&#8221; background_enable_image=&#8221;off&#8221; custom_padding=&#8221;10vw|0px|140px|0px|false|false&#8221; 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header_2_text_shadow_color__hover_enabled=&#8221;rgba(0,0,0,0.4)&#8221; sticky_enabled=&#8221;0&#8243;]Pfizer presented at a meeting of the AmericanChemical Society a potential anti-SARS-CoV-2 drug (PF-07321332), the firstorally administered coronavirus-specific protease inhibitor. CompoundPF-07321332 is currently in Phase 1 clinical trials and is the first orallyadministered compound that targets the main protease of SARS-CoV-2 virus, whichcauses COVID-19 disease. By inhibiting the main protease, PF-07321332 preventsthe virus from multiplying in the host cells. This compound is a covalentinhibitor that reacts with cysteine \u200b\u200bat the active site of the main protease.<\/p>\n<p>Because PF-07321332 can be taken orally, as atablet or capsule, it could be given outside hospitals if it proves to be safeand effective, which is a great advantage over intravenous drug formulations.Also, people who have been exposed to the SARS-CoV-2 virus could use this drugas a preventive measure.<\/p>\n<p>PF-07321332 is de novo developed drugduring the current SARS-CoV-2 virus pandemic. 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